首页> 外国专利> 4,5,6,7-TETRAHYDRO-L-BENZOTHIOPHENE MODULATORS OF RETINOIC ACID RECEPTOR RELATED (RAR) ORPHAN NUCLEAR RECEPTORS (RORS)

4,5,6,7-TETRAHYDRO-L-BENZOTHIOPHENE MODULATORS OF RETINOIC ACID RECEPTOR RELATED (RAR) ORPHAN NUCLEAR RECEPTORS (RORS)

机译:4,5,6,7-四氢-1-苯并噻吩调节剂的视黄酸受体相关(RAR)孤儿核受体(RORS)

摘要

The invention encompasses the novel class of compounds represented by the Formula (I), (II), (III) and (IV) below, which are modulators of RORγt:. The invention also encompasses pharmaceutical compositions which include the compounds shown above and methods of treating or preventing autoimmune diseases and antibody mediated rejection in a patient in need thereof.
机译:本发明包括以下内容(I),(II),(III)和(IV)所代表的新型化合物,其是RORγT的调节剂: 本发明还包括药物组合物,其包括上面所示的化合物以及治疗或预防适用于其患者中的自身免疫疾病和抗体介导的抑制的方法。

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