首页> 外国专利> NOVEL (HETEROCYCLE/TETRAHYDROPYRIDINE)-(PIPERAZINYL)-1-ALCANONE AND (HETEROCYCLE/DIHYDROPYRROLIDINE)-(PIPERAZINYL)-1-ALCANONE DERIVATIVES, AND USE THEREOF AS p75 INHIBITORS

NOVEL (HETEROCYCLE/TETRAHYDROPYRIDINE)-(PIPERAZINYL)-1-ALCANONE AND (HETEROCYCLE/DIHYDROPYRROLIDINE)-(PIPERAZINYL)-1-ALCANONE DERIVATIVES, AND USE THEREOF AS p75 INHIBITORS

机译:新型(杂环/四氢吡啶)-(哌嗪基)-1-Alcanone和(杂环/二氢吡啶基吡啶)-(哌嗪基)-1-Alcanone衍生物,并将其用作p75抑制剂

摘要

The disclosure relates to (heterocycle-tetrahydropyridine)(piperazinyl)-1-alkanone and (heterocycle-dihydropyrrolidine)(piperazinyl)-1-alkanone derivatives of formula (I):; embedded image ;wherein A, B, m, n, W, and R2 are as defined in the disclosure; to the methods of preparing said derivatives, and to the therapeutic uses thereof.
机译:本发明涉及式(I)的(杂环-四氢吡啶)(哌嗪基)-1-烷酮和(杂环-二氢吡咯烷)(哌嗪基)-1-烷酮衍生物: “嵌入式图像” ;其中,A,B,m,n,W和R2如本发明所定义;制备所述衍生物的方法及其治疗用途。

著录项

  • 公开/公告号US2012245150A1

    专利类型

  • 公开/公告日2012-09-27

    原文格式PDF

  • 申请/专利号US201213490905

  • 申请日2012-06-07

  • 分类号A61K31/496;A61K31/497;C07D487/08;A61K31/506;A61K31/444;C07D405/14;C07D401/14;C07D495/04;A61K31/551;A61K31/501;C07D417/14;A61P25/28;A61P25/08;A61P25/16;A61P25/18;A61P25/24;A61P25;A61P9;A61P9/10;A61P25/02;A61P27/02;A61P27/06;A61P17/14;A61P1/18;A61P1/16;A61P35;A61P35/04;A61P35/02;A61P11;A61P11/06;A61P37/08;A61P29;A61P37;A61P19/02;A61P17/06;A61P19/08;A61P19/10;C07D409/14;

  • 国家 US

  • 入库时间 2022-08-21 17:34:09

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