Copper-Catalyzed Oxidative -Ketoacylations of Sulfoximines with Aryl Methyl Ketones and Dioxygen as Terminal Oxidant

摘要

An efficient copper-catalyzed C-H/N-H bond functionalization for the synthesis of -keto-N-acyl sulfoximines from aryl methyl ketones and NH-sulfoximines with molecular oxygen as terminal oxidant has been developed.