机译:(R)-N-(3-(7-甲基-1H-吲唑-5-基)-1-(4-(1-甲基哌啶-4-基)-1-氧代丙烷-2-基)-4的发现 - 4 - (2-oxo-1,2-二氢喹啉-3-基)哌啶-1-甲酰胺(BMS-742413):具有优异的安全型材,用于通过鼻内递送治疗偏头痛的优异安全型材
Department of Molecular Sciences and Candidate Optimization Bristol-Myers Squibb RandD 5 Research;
Department of Molecular Sciences and Candidate Optimization Bristol-Myers Squibb RandD 5 Research;
Department of Neuroscience Discovery Biology Bristol-Myers Squibb RandD 5 Research Parkway;
Department of Neuroscience Discovery Biology Bristol-Myers Squibb RandD 5 Research Parkway;
Department of Neuroscience Discovery Biology Bristol-Myers Squibb RandD 5 Research Parkway;
Department of Neuroscience Discovery Biology Bristol-Myers Squibb RandD 5 Research Parkway;
Department of Neuroscience Discovery Biology Bristol-Myers Squibb RandD 5 Research Parkway;
Department of Neuroscience Discovery Biology Bristol-Myers Squibb RandD 5 Research Parkway;
Department of Molecular Sciences and Candidate Optimization Bristol-Myers Squibb RandD 5 Research;
Department of Molecular Sciences and Candidate Optimization Bristol-Myers Squibb RandD 5 Research;
Department of Molecular Sciences and Candidate Optimization Bristol-Myers Squibb RandD 5 Research;
Department of Molecular Sciences and Candidate Optimization Bristol-Myers Squibb RandD 5 Research;
Department of Molecular Sciences and Candidate Optimization Bristol-Myers Squibb RandD 5 Research;
Department of Molecular Sciences and Candidate Optimization Bristol-Myers Squibb RandD 5 Research;
Department of Molecular Sciences and Candidate Optimization Bristol-Myers Squibb RandD 5 Research;
Department of Molecular Sciences and Candidate Optimization Bristol-Myers Squibb RandD 5 Research;
Department of Molecular Sciences and Candidate Optimization Bristol-Myers Squibb RandD 5 Research;
Department of Molecular Sciences and Candidate Optimization Bristol-Myers Squibb RandD 5 Research;
CGRP receptor antagonist for intranasal delivery;
机译:(R)-N-(3-(7-甲基-1H-吲唑-5-基)-1-(4-(1-甲基哌啶-4-基)-1-氧代丙烷-2-基)-4的发现 - 4 - (2-oxo-1,2-二氢喹啉-3-基)哌啶-1-甲酰胺(BMS-742413):具有优异的安全型材,用于通过鼻内递送治疗偏头痛的优异安全型材
机译:基于结构的N - ((R)-3-(7-甲基-1H-吲唑-5-基)-1-氧代-1-((((s)-1-氧代-3-(哌啶 - 4-基)-1-(4-(吡啶-4-基)哌嗪-1-基)丙烷-2-基)氨基)丙酮-2-基)-2' -oxO-1',2'-DiHyDroSpiro [哌啶-4,4'-吡啶[2,3-D] [1,3]恶嗪] -1-甲酰胺(HTL22562):对偏头痛的急性治疗急性治疗的降钙素基因相关肽受体拮抗剂
机译:N-(((2H-Tetrazol-5-yl)methyl)-4-((R)-1-((5r,8R)-8-(叔丁基)-3-(3,5-二氯苯基)- 2-氧代-1,4-二氮杂螺并[4.5] dec-3-en-1-基)-4,4-二甲基戊基)苯甲酰胺(SCH 900822):有效的选择性胰高血糖素受体拮抗剂
机译:1-发现(4-(4- propionylpiperazin -1-基)-3-(三氟甲基)苯基)-9-(喹啉-3-基)苯并h 16萘啶-2(1H) - 一个作为雷帕霉素的高度有效的选择性的哺乳动物靶标(mTOR)抑制剂用于治疗癌症的治疗
机译:有效的口服生物可利用的降钙素基因相关的肽受体拮抗剂用于治疗偏头痛:发现n - (3r,6s)-6-(2,3-二氟苯基)-2-氧代-1-(2,2,2 - 三氟乙基)亚己己-3-基 -4-(2-氧代-2,3-二氢-1H-咪唑吡啶-1-基)哌啶-1-甲酰胺(MK-0974)