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机译:简单的四氢异喹啉是有效和选择性的κ阿片类受体拮抗剂
Research Triangle Institute PO Box 12194 Research Triangle Park North Carolina 27709-2194 United States;
Research Triangle Institute PO Box 12194 Research Triangle Park North Carolina 27709-2194 United States;
Research Triangle Institute PO Box 12194 Research Triangle Park North Carolina 27709-2194 United States;
Research Triangle Institute PO Box 12194 Research Triangle Park North Carolina 27709-2194 United States;
Research Triangle Institute PO Box 12194 Research Triangle Park North Carolina 27709-2194 United States;
Research Triangle Institute PO Box 12194 Research Triangle Park North Carolina 27709-2194 United States;
Research Triangle Institute PO Box 12194 Research Triangle Park North Carolina 27709-2194 United States;
Research Triangle Institute PO Box 12194 Research Triangle Park North Carolina 27709-2194 United States;
functional assays; JDTic; kappa opioid receptor antagonists; Opioid receptor; tetrahydroisoquinoline;
机译:简单的四氢异喹啉是有效和选择性的κ阿片类受体拮抗剂
机译:铅化合物(3R)-N-[1R)-1-(环己基甲基)-2-甲基丙基] -2-羟基-1,2,3,4-四氢异喹啉-3-甲基甲酰胺( CDTIC)
机译:(2S,3R)β-甲基-2',6'-二甲基肌氨酸-L-四氢异喹啉-3-羧酸[(2S,3R)TMT-L-Tic-OH]是一种有效的选择性δ-阿片受体拮抗剂老鼠的大脑
机译:kappa阿片受体拮抗剂的有效达氏菌的发展
机译:合成Salvinorin支架以开发潜在的止痛药和选择性,有效的阿片样物质配体
机译:铅化合物(3R)-7-羟基-N-(1S)-2-甲基-1-(哌啶-1-基甲基)丙基 -1234-的强选择性四氢异喹啉κ阿片受体拮抗剂四氢异喹啉-3-羧酰胺(PDTic)
机译:有效和选择性四羟基异喹啉kappa阿片受体铅化合物(3r)n 1r)1-(环己基甲基)-2-甲基丙基 -7-羟基-1,2,3,4-四氢异喹啉-3-甲酰胺(Cdtic)
机译:激活阿片受体主要介导Dadle的抗惊厥作用:U受体拮抗剂之间的相互作用