机译:AM-6226的发现:一种有效和口头生物可利用的GPR40完全激动剂,在非人的灵长类动物中显示出疗效
Department of Medicinal Chemistry Amgen Discovery Research One Amgen Center Drive;
Department of Medicinal Chemistry Amgen Discovery Research One Amgen Center Drive;
Department of Medicinal Chemistry Amgen Discovery Research One Amgen Center Drive;
Department of Medicinal Chemistry Amgen Discovery Research One Amgen Center Drive;
Department of Medicinal Chemistry Amgen Discovery Research One Amgen Center Drive;
Department of Medicinal Chemistry Amgen Discovery Research One Amgen Center Drive;
Department of Medicinal Chemistry Amgen Discovery Research One Amgen Center Drive;
Department of Medicinal Chemistry Amgen Discovery Research One Amgen Center Drive;
Department of Medicinal Chemistry Amgen Discovery Research One Amgen Center Drive;
Department of Medicinal Chemistry Amgen Discovery Research One Amgen Center Drive;
Department of Medicinal Chemistry Amgen Discovery Research One Amgen Center Drive;
Department of Medicinal Chemistry Amgen Discovery Research One Amgen Center Drive;
Department of Medicinal Chemistry Amgen Discovery Research One Amgen Center Drive;
AM-1638; AM-6226; AMG 837; FFA1; full agonist; GPR40; insulin secretagogue;
机译:AM-6226的发现:一种有效和口头生物可利用的GPR40完全激动剂,在非人的灵长类动物中显示出疗效
机译:DS-1558的发现:一种有效且口服生物利用的GPR40激动剂
机译:发现三氟甲基(嘧啶-2-基)氮杂环丁烷-2-羧酰胺为有效的,口服生物利用的TGR5(GPBAR1)激动剂:结构-活性关系,铅优化和慢性体内功效
机译:发现有效的MMCLR激动剂,具有延长人黑素细胞的长期活动
机译:具有有效抗疟疾活性的口服生物可利用的4(1H)-喹诺酮和1,2,3,4-Tetrahydroacridin-9(10H)-ones的开发
机译:AM-6226的发现:有效且可口服的生物利用度GPR40全激动剂可在非人类灵长类动物中显示功效
机译:DS-1558的发现:一种有效和口服的生物可利用的GPR40激动剂
机译:超抗原诱导的细胞因子从全血细胞培养中释放,作为非人灵长类动物口服给药后药物功效的功能测量