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18th European Symposium on Radiopharmacy and Radiopharmaceuticals

机译:第十八届欧洲放射性药物和放射性药物专题讨论会

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OP03 Selective extraction of medically-related radionuclides from proton-irradiated thorium targets V. Radchenko, J.W. Engle, C. Roy, J. Griswold, M.F. Nortier, E.R. Birnbaum, M. Brugh, S. Mirzadeh, K. D. John, M.E. Fassbender OP04 Comparison of [68Ga]FSC(succ-RGD)3 and [68Ga]NODAGA-RGD for PET imaging of αvβ3 integrin expression Chuangyan Zhai, Gerben M. Franssen, Milos Petrik, Peter Laverman, Clemens Decristoforo OP05 A new NPY-Y1R targeting peptide for breast cancer PET imaging Ait-Mohand Samia, Dumulon-Perreault Véronique, Guérin Brigitte OP06 The influence of multivalency on CCK 2 receptor targeting D. Summer, A. Kroess, C. Rangger, H. Haas, P. Laverman, F. Gerben, E. von Guggenberg, C.Decristoforo OP07 SPECT Imaging of αvβ3 Expression by [99mTc(N)PNP43]- Bifunctional Chimeric RGD Peptide not Cross-Reacting with αvβ5 Cristina Bolzati, Nicola Salvarese, Fiorenzo Refosco, Laura Meléndez-Alafort, Debora Carpanese, Antonio Rosato, Michele Saviano, Annarita Del Gatto, Daniela Comegna, Laura Zaccaro OP09 New dienophiles for the inverse-electron-demand Diels-Alder reaction and for pretargeted PET imaging Emilie Billaud, Muneer Ahamed, Frederik Cleeren, Elnaz Shahbazali, Tim No?l, Volker Hessel, Alfons Verbruggen and Guy Bormans OP10 New complexing agent for Al18F-labelling of heat-sensitive biomolecules: Synthesis and preclinical evaluation of Al18F-RESCA1-HAS Cleeren F, Lecina J, Koole M, Verbruggen A and Bormans G OP11 A novel versatile precursor efficient for F-18 radiolabelling via click-chemistry B. Lugatoa, S. Stucchia, E.A. Turollaa, L. Giulianoa, S.Toddea, P. Ferraboschib OP12 A general applicable method to quantify unidentified UV impurities in radiopharmaceuticals R.P. Klok, M.P.J. Mooijer, N.H. Hendrikse, A.D. Windhorst OP13 Development of [18F]Fluoro-C-glycosides to radiolabel peptides Collet C., Petry N., Chrétien F., Karcher G., Pellegrini-Mo?se N., Lamandé-Langle S. OP14 A Microfluidic Approach for the 68Ga-labeling of PSMAHBED-CC and NODAGA-RGD Sarah Pfaff, Cecile Philippe, Markus Mitterhauser, Marcus Hacker, Wolfgang Wadsak OP16 Surprising reactivity of astatine in the nucleophilic substitution of aryliodonium salts: application to the radiolabeling of antibodies Fran?ois Guérard, Yong-Sok Lee, Sébastien Gouard, Kwamena Baidoo, Cyrille Alliot, Michel Chérel, Martin W. Brechbiel, Jean-Fran?ois Gestin OP17 64Cu-NOTA-pertuzumab F(ab')2 fragments, a second-generation probe for PET imaging of the response of HER2-positive breast cancer to trastuzumab (Herceptin) Lam K, Chan C, Reilly RM OP18 Development of radiohalogenated analogues of a avb6-specific peptide for high LET particle emitter targeted radionuclide therapy of cancer Salomé Paillas, John Marshall, Jean-Pierre Pouget, Jane Sosabowski OP19 Ligand Specific Efficiency (LSE) as a guide in tracer optimization Emmanuelle Briard, Yves P. Auberson, John Reilly, Mark Healy, David Sykes OP23 The radiosynthesis of an 18F-labeled triglyceride, developed to visualize and quantify brown adipose tissue activity Andreas Paulus, Wouter van Marken Lichtenbelt,Felix Mottaghy, Matthias Bauwens OP24 Influence of the fluorescent dye on the tumor targeting properties of dual-labeled HBED-CC based PSMA inhibitors Baranski, Ann-Christin, Sch?fer, Martin, Bauder-Wüst, Ulrike, Haberkorn, Uwe, Eder, Matthias, Kopka, Klaus OP25 [18F]MEL050 as a melanin PET tracer : fully automated radiosynthesis and evaluation for the detection of pigmented melanoma in mice pulmonary metastases Chaussard M, Hosten B, Vignal N, Tsoupko-Sitnikov V, Hernio N, Hontonnou F, Merlet P, Poyet JL, Sarda-Mantel L, Rizzo-Padoin N OP26 Design and Preclinical Evaluation of Novel Radiofluorinated PSMA Targeting Ligands Based on PSMA-617 J. Cardinale, M. Sch?fer, M. Bene?ová, U. Bauder-Wüst, O. Seibert, F. Giesel, U. Haberkorn, M. Eder, K. Kopka OP27 A novel radiolabeled peptide for PET imaging of prostate cancer: 64Cu-DOTHA2-PEG-RM26 Mansour Nematallah, Paquette Michel, Ait-Mohand Samia, Dumulon-Perreault Véronique, Lecomte Roger, Guérin Brigitte OP29 Biodistribution of [18F]Amylovis?, a new radiotracer PET imaging of β-amyloid plaques Fernandez-Maza L, Rivera-Marrero S, Prats Capote A, Parrado-Gallego A, Fernandez-Gomez I, Balcerzyk M, Sablon-Carrazana M, Perera-Pintado A, Merceron-Martinez D, Acosta-Medina E, Rodriguez-Tanty C OP30 Synthesis and preclinical evaluation of [11C]-BA1 PET tracer for the imaging of CSF-1R Bala Attili, Muneer Ahamed, Guy Bormans OP31 In vivo imaging of the MCHR1 in the ventricular system via [18F]FE@SNAP C. Philippe, M. Zeilinger, T. Scherer, C. Fürnsinn, M. Dumanic, W. Wadsak, M. Hacker, M. Mitterhauser OP32 Synthesis of the first carbon-11 labelled P2Y12 receptor antagonist for imaging the anti-inflammatory phenotype of activated microglia B. Janssen, D.J. Vugts, G.T. Molenaar, U. Funke, P.S. Kruijer, F. Dollé, G. Bormans, A.A. Lammertsma, A.D. Windhorst OP33 Radiosynthesis of a selective HDAC6 inhibitor [11C]KB631 and i
机译:OP03从质子辐照的targets靶上选择性提取医学相关的放射性核素V. Radchenko,J.W. Engle,C.Roy,J.Griswold,M.F。 Nortier,ER Birnbaum,M。Brugh,S。Mirzadeh,KD John,ME Fassbender OP04对[68Ga] FSC(succ-RGD)3和[68Ga] NODAGA-RGD进行αvβ3整合素表达的PET成像的比较Chuangyan Zhai,Gerben M 。Franssen,Milos Petrik,Peter Laverman,Clemens Decristoforo OP05用于乳腺癌PET成像的新型NPY-Y1R靶向肽Ait-Mohand Samia,Dumulon-PerreaultVéronique,GuérinBrigitte OP06多价对CCK 2受体靶向D的影响。 A. Kroess,C。Rangger,H。Haas,P。Laverman,F。Gerben,E。von Guggenberg,C.Decristoforo OP07 SPECT通过[99mTc(N)PNP43]-双功能嵌合RGD肽对αvβ3表达的成像与αvβ5克里斯蒂娜·博尔扎蒂(Cristina Bolzati),尼古拉·萨尔瓦雷斯(Nicola Salvarese),菲奥伦佐·雷福斯科(Fiorenzo Refosco),劳拉·梅伦德斯·阿拉福特(LauraMeléndez-Alafort),黛博拉·卡拉帕尼斯(Antonio Rosato),米歇尔·萨维亚诺(Michele Saviano),安娜里塔·德尔·加托(Daniela Comegna),劳拉·扎卡罗OP09反应用于预先定位的PET成像Emilie Billaud,Muneer Ahamed,F rederik Cleeren,Elnaz Shahbazali,Tim No?l,Volker Hessel,Alfons Verbruggen和Guy Bormans OP10用于热敏生物分子Al18F标记的新型络合剂:Al18F-RESCA1-HAS的合成和临床前评价Cleeren F,Lecina J,Koole M,Verbruggen A和Bormans G OP11一种新颖的通用前体,可通过点击化学B有效用于F-18放射性标记。Lugatoa,S。Stucchia,EA Turollaa,L.Giuliaona,S.Toddea,P.Ferraboschib OP12一种通用的定量放射性药物中未鉴定的UV杂质的方法R.P. Klok,M.P.J. Mooijer,NH Hendrikse,AD Windhorst OP13 [ 18 F]氟-C-糖苷开发为放射性标记肽的方法Collet C.,Petry N.,ChrétienF.,Karcher G.,Pellegrini-Mo?se N.,Lamandé-LangleS. OP14用于PSMAHBED-CC和NODAGA-RGD 68Ga标记的微流控方法Sarah Pfaff,Cecile Philippe,Markus Mitterhauser,Marcus Hacker,Wolfgang Wadsak OP16 ine素在亲核取代芳草醚中的惊人反应性盐:在抗体放射标记中的应用Fran?oisGuérard,Lee-Sok Lee,SébastienGouard,Kwamena Baidoo,Cyrille Alliot,MichelChérel,Martin W. Brechbiel,Jean-Fran?ois Gestin OP17 64 Cu-NOTA-pertuzumab F(ab') 2 片段,用于PET成像的HER2阳性乳腺癌对曲妥珠单抗(赫赛汀)反应的第二代探针Lam K,Chan C,Reilly RM OP18开发用于高LET粒子发射器靶向的放射性核素治疗癌症的avb6特异性肽的放射性卤代类似物SaloméPaillas,John Marshall,Jean-Pierre Pouget,Jane Sosabowski OP19配体比效率(LSE)作为示踪剂优化的指南Emmanuelle Briard,Yves P.Auberson,John Reilly,Mark Healy,David Sykes OP23标记18F的放射性合成甘油三酸酯,开发用于可视化和量化棕色脂肪组织的活性Andreas Paulus,Wouter van Marken Lichtenbelt,Felix Mottaghy,Matthias Bauwens OP24荧光染料对基于双标记HBED-CC的PSMA抑制剂靶向肿瘤的特性的影响Baranski,Ann-Christin ,Sch?fer,Martin,Bauder-Wüst,Ulrike,Haberkorn,Uwe,Eder,Matthias,Kopka,Klaus OP25 [18F] MEL050作为黑色素PET示踪剂:全自动放射合成和评估小鼠肺转移中色素性黑色素瘤的检测Chaussard M,Hosten B,Vignal N,Tsoupko-Sitnikov V,Hernio N,Hontonnou F,Merlet P,Poyet JL,Sarda-Mantel L,Rizzo-Padoin N OP26新型放射性氟化PSMA靶标的设计和临床前评估基于PSMA-617的配体J. Cardinale,M。Sch?fer,M。Bene?ová,U。Bauder-Wüst,O。Seibert,F。Giesel,U。Haberkorn,M。Eder,K。Kopka OP27 A用于前列腺癌PET成像的新型放射性标记肽:64Cu-DOTHA2-PEG-RM26 Mansour Nematallah,Paquette Michel,Ait-Mohand Samia,Dumulon-PerreaultVéronique,Lecomte Roger,GuérinBrigitte OP29 [ 18 的生物分布F] Amylovis ?,一种新的放射性示踪剂PET成像,用于β-淀粉样蛋白斑Fernandez-Maza L,Rivera-Marrero S,Prats Capote A,Parrado-Gallego A,Fernandez-Gomez I,Balcerzyk M,Sablon-Carrazana M,Perera-Pintado A,Merceron-Martinez D,Acosta-Medina E,Rodriguez-Tanty C OP30 [11C] -BA1 PET示踪剂的合成和临床前评价,用于CSF-1R Bala Attili,Muneer Ahamed,Guy Bormans OP31的体内成像C. Philippe,M. Zeilinger,T. Scherer,C.Fürnsinn,M.Dumanic,W.Wadsak,M. Hacker,M.Mitterhauser OP32通过[18F] FE @ SNAP在心室系统中生成MCHR1。 11标签ed P2Y12受体拮抗剂,用于对活化的小胶质细胞B的抗炎表型进行成像。Janssen,D.J. Vugts,G.T.美国丰克大学Molenaar Kruijer,F.Dollé,G.Bormans,A.A。 Lammertsma,A.D. Windhorst OP33选择性HDAC6抑制剂[11C] KB631和i的放射合成

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