首页> 外国专利> TRICYCLIC COMPOUNDS HAVING ACTIVITY SPECIFIC FOR INTEGRINS, PARTICULARLY αvβ3 INTEGRINS, METHOD FOR PREPARING SAME, INTERMEDIATES THEREFOR, USE OF SAID COMPOUNDS AS DRUGS, AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME

TRICYCLIC COMPOUNDS HAVING ACTIVITY SPECIFIC FOR INTEGRINS, PARTICULARLY αvβ3 INTEGRINS, METHOD FOR PREPARING SAME, INTERMEDIATES THEREFOR, USE OF SAID COMPOUNDS AS DRUGS, AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME

机译:三环化合物具有特定于整合素的活性,尤其是αvβ3整合素,其制备方法,中间体,将上述化合物用作药物的药物以及包含相同化合物的药物组合物

摘要

Compounds of formula (I), wherein R1, R2, R3, R4, R5 and G are as defined in the description and the dotted lines indicate an optional second bond, as well as the acid, base and ester addition salts thereof, a method for preparing said compounds, intermediates therefor, the use of said compounds as drugs, and pharmaceutical compositions containing same, are disclosed.
机译:其中R1,R2,R3,R4,R5和G如说明书中所定义且虚线表示任选的第二键的式(I)化合物及其酸,碱和酯加成盐,一种方法为了制备所述化合物,公开了其中间体,所述化合物作为药物的用途以及包含所述化合物的药物组合物。

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