where R1 and R2 each means independently each of other mono- or di-substituted residues with A, OH, OA, phenylmethoxy, -O-(CH2)n-O-, NH2, NHAc, NAAc, NHSO2A, fluorine or chlorine atom, phenyl; X means O, S or SO2; m = 1; n = 2; A is C1-6-atoms; Ac is C1-4-alkanoyl and also their physiologically acceptable salts that effect on CNS being damping effect preferably. EFFECT: improved method of synthesis and preparing, central effects. 11 cl, 1 tbl, 21 ex"/>
4-ARYLOXY- OR 4-ARYLTHIOPIPERIDINE DERIVATIVES, METHODS OF THEIR SYNTHESIS, PHARMACEUTICAL COMPOSITION CONTAINING ON SAID AND METHOD OF ITS PREPARING
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4-ARYLOXY- OR 4-ARYLTHIOPIPERIDINE DERIVATIVES, METHODS OF THEIR SYNTHESIS, PHARMACEUTICAL COMPOSITION CONTAINING ON SAID AND METHOD OF ITS PREPARING
4-ARYLOXY- OR 4-ARYLTHIOPIPERIDINE DERIVATIVES, METHODS OF THEIR SYNTHESIS, PHARMACEUTICAL COMPOSITION CONTAINING ON SAID AND METHOD OF ITS PREPARING
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机译：4-芳氧或4-芳硫哌啶衍生物，其合成方法，包含上述成分的药物成分及其制备方法
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FIELD: organic chemistry, pharmacy. SUBSTANCE: invention relates to 4-aryloxy- or 4-arylthio- -piperidine derivatives of the formula (I) where R1 and R2 each means independently each of other mono- or di-substituted residues with A, OH, OA, phenylmethoxy, -O-(CH2)n-O-, NH2, NHAc, NAAc, NHSO2A, fluorine or chlorine atom, phenyl; X means O, S or SO2; m = 1; n = 2; A is C1-6-atoms; Ac is C1-4-alkanoyl and also their physiologically acceptable salts that effect on CNS being damping effect preferably. EFFECT: improved method of synthesis and preparing, central effects. 11 cl, 1 tbl, 21 ex
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机译：领域：有机化学，药学。物质：本发明涉及式（I）的4-芳氧基-或4-芳硫基-哌啶衍生物<图像文件=“ 00000001.GIF” he =“ 26” imgContent =“ undefined” imgFormat =“ GIF” wi =“ 67“ />，其中R 1 和R 2 分别独立地表示具有A，OH，OA，苯基甲氧基，-O-（ CH 2 ） n -O-，NH 2 ，NHAc，NAAc，NHSO 2 A，氟或氯原子，苯基; X表示O，S或SO 2 ; m = 1; n = 2; A是C 1-6 原子; Ac是C 1-4 -烷酰基，并且它们对CNS起作用的生理上可接受的盐优选为阻尼作用。效果：改进的合成和制备方法，主要作用。 11厘升，1汤匙，21前
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