首页> 外国专利> Derivatives of 3,4 - substituted aryl or heteroaryl dihydro anthracene or benzo 1,2-g - chrom - 3 - eno substituted aryl or heteroaryl or benzo 1,2-g - thiocrom-3-ene and benzo 1, 2-g -1,2- dihydroquinoline having retinoid antagonist or inverse retinoid agonist biological activity

Derivatives of 3,4 - substituted aryl or heteroaryl dihydro anthracene or benzo 1,2-g - chrom - 3 - eno substituted aryl or heteroaryl or benzo 1,2-g - thiocrom-3-ene and benzo 1, 2-g -1,2- dihydroquinoline having retinoid antagonist or inverse retinoid agonist biological activity

机译:3,4-取代的芳基或杂芳基二氢蒽或苯并[1,2-g]的衍生物-铬3-烯基取代的芳基或杂芳基或苯并[1,2-g]-硫代crom-3-ene和苯并[1] ,2 g] -1,2-二氢喹啉具有类维生素A拮抗剂或类维生素A激动剂反向生物活性

摘要

Invention Patent: B "REPLACED 3,4-DIHYDROANTHRACENO ARILA OR HETEROARILLA OR BENZO [1,2-g] -CROM-3-ENO SUBSTITUTE ARILA OR HETEROARILLA, BENZO [1.2-g] -TIOCROM-3- ENO AND BENZO [1,2-g] -1-2-DIHYDROQUINOLIN HAVING BIOLOGICAL ACTIVITY TYPE OF RETINOID ANTAGONIST OR REVERSE RETINOID AGONIST "D. Compounds of formula (1), where the symbols have the meanings defined in the specification, have biological activity like retinoid, retinoid antagonist and / or inverse retinoid agonist.
机译:发明专利:“取代了3,4-二氢蒽环杂芳基或杂芳基或苯并[1,2-g] -CROM-3-ENO取代杂芳基杂芳基或苯并[1.2-g] -TIOCROM-3-ENO和苯并具有生物活性类型的类视黄酸拮抗剂或反向类视黄酸激动剂“ ”​​的[1,2-g] -1-2-二氢喹诺灵。其中符号具有说明书中定义的含义的式(1)化合物具有生物活性,如类维生素A,类维生素A拮抗剂和/或类维生素A反向激动剂。

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