首页> 外国专利> ANTIGONIST COMBINATION THERAPY OF ALDOSTERONE EPOXY-STEROID AND ANGIOTENSIN II ANTAGONIST FOR THE TREATMENT OF CONGESTIVE CARDIAC FAILURE.

ANTIGONIST COMBINATION THERAPY OF ALDOSTERONE EPOXY-STEROID AND ANGIOTENSIN II ANTAGONIST FOR THE TREATMENT OF CONGESTIVE CARDIAC FAILURE.

机译:醛固酮环氧-类固醇和血管紧张素II拮抗剂的拮抗剂联合治疗,用于治疗充血性心力衰竭。

摘要

A COMBINATION THERAPY THAT INCLUDES A THERAPEUTICALLY EFFECTIVE AMOUNT OF AN EFFECTIVE ALDOSTERONE RECEIVER ANTAGONIST OF AN ANTIGONIST OF THE ANGIOTENSIN II RECEIVER ANTAGONIST FOR THE TREATMENT OF CIRCULATORY CIRCULAR CIRCULAR DISTRIBUTIONS, CARDINES, CARBON CIRCULAR DISCUSSIONS ASCITES. THE PREFERRED ANTAGONISTS OF THE ANGIOTENSIN II RECEIVER ARE THOSE COMPOUNDS THAT HAVE A HIGH POWER AND BIODISPONIBILITY AND THAT ARE CHARACTERIZED BY POSSESSING AN IMIDAZOL OR TRIAZOL GROUP JOINED TO A BIFENILMETILO OR PIRIDINIL. THE ANTAGONISTS OF THE ALDOSTERONE EPOXI RECEIVER ARE SPIROXAN STEROID COMPOUNDS OR THE PRESENCE OF AN EPOXI PORTION REPLACED IN 9 AL}, 11 AL}. A PREFERRED COMBINATION THERAPY INCLUDES THE ANGIOTENSIN II RECEIVER ANTAGONIST 5 TETRAZOL AND THE ALDOSTERONE EPOXIMEXRENONE RECEIVER ANTAGONIST.
机译:包含治疗性有效量的有效量的阿尔度孕酮受体拮抗剂和抗血管紧张素II受体拮抗剂的组合疗法,用于治疗循环圆环分布,心血管分布。血管紧张素II受体的首选拮抗剂是具有高功率和生物亲和性的化合物,其特征在于具有与二苯甲腈或吡喹啉联用的咪唑或三唑基团。醛固酮环氧化合物受体的拮抗剂是吡咯烷酮类固醇化合物或存在于9 AL 1 1,11 AL 1中的环氧化合物部分。优选的组合治疗包括血管紧张素II受体拮抗剂5四唑和醛固酮表二氧戊烯酮受体拮抗剂。

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