首页> 外国专利> crystalline polymorph, composition, methods of preparing the polymorphic form of bazedoxifene acetate, treating a mammal having a disease or syndrome associated with estrogen deficiency or excess estrogen, and with abnormal proliferation or development of endometrial tissues, breast cancer in a mammal, and a postmenopausal woman for one or more vasomotor disorders, lowering cholesterol in a mammal, and inhibiting bone loss in a mammal, and, form the crystalline polymorph of bazedoxifene acetate

crystalline polymorph, composition, methods of preparing the polymorphic form of bazedoxifene acetate, treating a mammal having a disease or syndrome associated with estrogen deficiency or excess estrogen, and with abnormal proliferation or development of endometrial tissues, breast cancer in a mammal, and a postmenopausal woman for one or more vasomotor disorders, lowering cholesterol in a mammal, and inhibiting bone loss in a mammal, and, form the crystalline polymorph of bazedoxifene acetate

机译:结晶多晶型物,组合物,乙酸巴多昔芬乙酸酯的多晶型物的制备方法,治疗患有与雌激素缺乏或雌激素过多有关的疾病或综合征,子宫内膜组织异常增生或发育的哺乳动物,哺乳动物的乳腺癌以及绝经后的方法一种或多种血管舒缩性疾病的女性,降低哺乳动物的胆固醇水平,抑制哺乳动物的骨质流失,并形成醋酸巴多昔芬醋酸盐的结晶多晶型物

摘要

CRYSTALLINE POLYMORPH, COMPOSITION, METHODS OF PREPARING FOR THE BAZEDOXYPHEN ACETATE POLYMORPHIC, TREATING A MAMMER WITH A DISEASE OR SYNDROME ASSOCIATED WITH ESTROGEN DEFENSE OR EXCESSION CUT MAMMALIAN, AND A POST-MENOPAUSAL WOMAN FOR ONE OR VARIOUS VASOMOTOR DISORDERS, TO LOWER CHOLESTEROL IN A MAMMER, AND TO INHIBIT BONE LOSS IN A MAMMER, AND FORM THE CRYSTALLINE POLYMORPH OF BAZEDOXYPHYPHENE. The present invention relates to a crystalline polymorph of bazedoxifene acetate, compositions containing the same, their preparations, and their uses.
机译:结晶多态性,组成,制备乙酸巴多巴多酚的方法,治疗伴有雌激素防御或疾病的哺乳动物或伴有疾病或综合征的哺乳动物,以及绝经后的哺乳动物经口为一个或一个时期的绝经期妇女。 ,并阻止其在骨骼中的流失,并形成重金属卟啉的结晶多晶。本发明涉及乙酸巴多昔芬乙酸盐的结晶多晶型物,包含其的组合物,其制备方法及其用途。

著录项

  • 公开/公告号BRPI0509191A

    专利类型

  • 公开/公告日2007-09-25

    原文格式PDF

  • 申请/专利权人 WYETH;

    申请/专利号BR2005PI09191

  • 申请日2005-04-06

  • 分类号C07D209/12;A61K31/404;A61K31/55;A61P5/30;C07D403/12;

  • 国家 BR

  • 入库时间 2022-08-21 20:59:22

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