首页> 外国专利> 4-ä'3- (SULFONYLAMINO) PHENYLÜ'1- (CYCLYMETHYL) PIPERIDINE-4-YLIDENEUMETHYLENEZAMIDE DERIVATIVES AS DELTA OPIOID RECEPTOR LIGANDS FOR THE TREATMENT OF PAIN, FEARING STATE AND FUNCTIONAL GASTROINTESTINAL ILLNESSES

4-ä'3- (SULFONYLAMINO) PHENYLÜ'1- (CYCLYMETHYL) PIPERIDINE-4-YLIDENEUMETHYLENEZAMIDE DERIVATIVES AS DELTA OPIOID RECEPTOR LIGANDS FOR THE TREATMENT OF PAIN, FEARING STATE AND FUNCTIONAL GASTROINTESTINAL ILLNESSES

机译:4-Δ'3-(磺酰胺基)苯'1-(环甲基)哌啶-4-亚乙基亚甲基乙酰胺衍生物作为阿片类阿片受体类药物治疗疼痛,恐惧状态和功能性胃肠道不适

摘要

Compounds of general formula: (I) wherein RSUP1/SUP, RSUP2/SUP, RSUP3/SUP, RSUP4 /SUPand RSUP5 /SUPare as defined in the specification, as well as salts, enantiomers thereof and pharmaceutical compositions including the compounds are prepared. They are useful in therapy, in particular in the management of pain.
机译:通式(I)的化合物,其中R 1 ,R 2 ,R 3 ,R 4 和R说明书中定义了 5 ,并制备了其盐,对映异构体和包括该化合物的药物组合物。它们可用于治疗,特别是在疼痛的治疗中。

著录项

  • 公开/公告号DE602004002933T2

    专利类型

  • 公开/公告日2007-09-06

    原文格式PDF

  • 申请/专利权人 ASTRAZENECA AB;

    申请/专利号DE20046002933T

  • 发明设计人

    申请日2004-01-13

  • 分类号C07D409/06;C07D405/06;C07D211/70;C07D401/06;C07D417/06;C07C311/08;A61K31/4436;A61K31/443;A61K31/44;A61K31/444;A61K31/4439;A61P25/04;

  • 国家 DE

  • 入库时间 2022-08-21 20:28:11

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