首页> 外国专利> METHODS FOR TREATING AT LEAST ONE CONDITION HAVING MT1 RECEPTOR, 5HT2B RECEPTOR, AND L-TYPE CALCIUM CHANNEL ACTIVITY.

METHODS FOR TREATING AT LEAST ONE CONDITION HAVING MT1 RECEPTOR, 5HT2B RECEPTOR, AND L-TYPE CALCIUM CHANNEL ACTIVITY.

机译:具有MT1受体,5HT2B受体和L型钙离子通道活性的至少一种条件的治疗方法。

摘要

The present invention is directed to methods comprising administering a composition comprising a therapeutically effective amount of (R)-verapamil, a derivative thereof, or a pharmaceutically acceptable salt thereof, wherein the composition treats, prevents and/or manages at least one condition having MT1 receptor, 5-HT2B receptor and L-type calcium channel activity and releases the (R)-verapamil, a derivative thereof or a pharmaceutically acceptable salt thereof to exhibit a co-primary activity on the MT1 receptor, the 5-HT2B receptor, and the L- type calcium channel.
机译:本发明涉及方法,该方法包括给予包含治疗有效量的(R)-维拉帕米,其衍生物或其药学上可接受的盐的组合物,其中该组合物治疗,预防和/或控制至少一种患有MT1的疾病受体,5-HT2B受体和L型钙通道活性,并释放(R)-维拉帕米,其衍生物或其药学上可接受的盐,以表现出对MT1受体,5-HT2B受体的共主要活性。 L型钙通道。

著录项

  • 公开/公告号MX2009000923A

    专利类型

  • 公开/公告日2009-03-09

    原文格式PDF

  • 申请/专利权人 AGI THERAPEUTICS RESEARCH LTD.;

    申请/专利号MX20090000923

  • 发明设计人 JOHN DEVANE;MARY MARTIN;JOHN KELLY;

    申请日2007-07-18

  • 分类号A61P25/06;A61K31/277;

  • 国家 MX

  • 入库时间 2022-08-21 19:26:27

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