首页> 外国专利> A NEW DERIVATIVE OF 1,4-BENZOTIAZEPINE-1,1-DIOXIDE WITH IMPROVED PROPERTIES, METHOD FOR ITS PRODUCTION, MEDICINE CONTAINING THE INDICATED COMPOUND AND ITS APPLICATION

A NEW DERIVATIVE OF 1,4-BENZOTIAZEPINE-1,1-DIOXIDE WITH IMPROVED PROPERTIES, METHOD FOR ITS PRODUCTION, MEDICINE CONTAINING THE INDICATED COMPOUND AND ITS APPLICATION

机译:一种具有改进性能的1,4-苯并二氮杂EP庚因-1,1-二氧化物的新衍生物,其制备方法,含该指示化合物的药物及其应用

摘要

1. The compound of formula A! ! and its pharmaceutically acceptable salts. ! 2. A drug containing a compound according to claim 1, to normalize lipid metabolism. ! 3. A drug containing a compound according to claim 1 and at least one additional biologically active substance, to normalize lipid metabolism. ! 4. The drug according to claim 3, characterized in that as an additional biologically active substance, it contains one or more compounds that normalize lipid metabolism. ! 5. The drug according to claim 3 or 4, characterized in that as an additional biologically active substance it contains one or more antidiabetic agents, hypoglycemic agents, anti-obesity drugs, appetite suppressants, HMGCoA reductase inhibitors, cholesterol resorption inhibitors , PPAR gamma agonists, PPAR alpha agonists, PPAR alpha / gamma agonists, fibrates, MTP inhibitors, CETP inhibitors, polymeric bile acid adsorbers, pathogens of LDL receptors, ACAT inhibitors, antioxidants, in lipoprotein lipase inhibitors, ATP-citrate lyase inhibitors, squalene synthetase inhibitors, lipoprotein (s) antagonists, lipase inhibitors, insulin, sulfonylureas, biguanides, meglitinides, thiazolidinediones, alpha-glucosidase-dependent, biologically active channel-dependent, biologically active cells, biologically active substances CART agonists, NPY agonists, cannabinoid receptor 1 antagonists, MCH receptor antagonists, MC4 agonists, orexin agonists, H3 agonists, TNF agonists, CRF agonists, CRF BP antagonists, GLP-1 derivatives, agonist urocortin ov, β3 agonists, MSH (chalk
机译:1.式A化合物! !及其药学上可接受的盐。 ! 2.一种药物,其包含根据权利要求1的化合物,以使脂质代谢正常化。 ! 3.一种药物,其包含根据权利要求1的化合物和至少一种另外的生物活性物质,以使脂质代谢正常化。 ! 4.根据权利要求3所述的药物,其特征在于,作为另外的生物活性物质,其包含使脂质代谢正常化的一种或多种化合物。 ! 5.根据权利要求3或4所述的药物,其特征在于,作为另外的生物活性物质,其包含一种或多种抗糖尿病药,降血糖药,抗肥胖药,食欲抑制剂,HMGCoA还原酶抑制剂,胆固醇吸收抑制剂,PPARγ激动剂。 ,PPARα激动剂,PPARα/γ激动剂,贝特类,MTP抑制剂,CETP抑制剂,聚合胆汁酸吸附剂,LDL受体病原体,ACAT抑制剂,抗氧化剂,脂蛋白脂肪酶抑制剂,ATP柠檬酸裂解酶抑制剂,角鲨烯合成酶抑制剂,脂蛋白(s)拮抗剂,脂肪酶抑制剂,胰岛素,磺酰脲类,双胍类,美格替宁,噻唑烷二酮,α-葡萄糖苷酶依赖性,生物活性通道依赖性,生物活性细胞,生物活性物质CART激动剂,NPY激动剂,大麻素受体1拮抗剂,MCH受体拮抗剂,MC4激动剂,orexin激动剂,H3激动剂,TNF激动剂,CRF激动剂,CRF BP anta激动剂,GLP-1衍生物,激动剂urocortin ov,β3激动剂,MSH(粉笔

著录项

相似文献

  • 专利
  • 外文文献
  • 中文文献
获取专利

客服邮箱:kefu@zhangqiaokeyan.com

京公网安备:11010802029741号 ICP备案号:京ICP备15016152号-6 六维联合信息科技 (北京) 有限公司©版权所有
  • 客服微信

  • 服务号