首页> 外国专利> n- (5-chlorosalicyl) -5-aminocaproic acid disodium salt form i, n- (5-salicyloyl) -8-aminocaprylic acid disodium salt monohydrate, n- (5- (5-salicyloyl) disodium salt monohydrate) chlorosalicyloyl) -5-aminocaproic acid, n- (5-salicoyloyl) -8-aminocaprylic acid disodium salt crystalline ethanol solvate, n- (5-chlorosalicyloyl) -5-aminocaproic acid disodium salt form iii, salt octahidrate n- (5-salicyloyl) -8-aminocaprylic acid disodium, n- (5-salicyloyl) -8-aminocaprylic acid disodium salt monohydrate, pharmaceutical composition, process for preparing n-disodium salt form i (5-salicyloyl) -8-aminocaprylic acid, process for preparing an n- (5-salicyloyl) -8-aminocaprylic acid disodium salt monoethanol solvate, process for preparing a 5-cnac octahidrate, process for preparing iv form n- (5-salicyloyl) -8-aminocaprylic acid disodium salt and process for preparing a mixture of the n- (5-salicyloyl) -8-aminocaprylic acid disodium salt forms i and iv

n- (5-chlorosalicyl) -5-aminocaproic acid disodium salt form i, n- (5-salicyloyl) -8-aminocaprylic acid disodium salt monohydrate, n- (5- (5-salicyloyl) disodium salt monohydrate) chlorosalicyloyl) -5-aminocaproic acid, n- (5-salicoyloyl) -8-aminocaprylic acid disodium salt crystalline ethanol solvate, n- (5-chlorosalicyloyl) -5-aminocaproic acid disodium salt form iii, salt octahidrate n- (5-salicyloyl) -8-aminocaprylic acid disodium, n- (5-salicyloyl) -8-aminocaprylic acid disodium salt monohydrate, pharmaceutical composition, process for preparing n-disodium salt form i (5-salicyloyl) -8-aminocaprylic acid, process for preparing an n- (5-salicyloyl) -8-aminocaprylic acid disodium salt monoethanol solvate, process for preparing a 5-cnac octahidrate, process for preparing iv form n- (5-salicyloyl) -8-aminocaprylic acid disodium salt and process for preparing a mixture of the n- (5-salicyloyl) -8-aminocaprylic acid disodium salt forms i and iv

机译:n-(5-氯水杨基)-5-氨基己酸二钠盐形式,n-(5-水杨酰基)-8-氨基辛酸二钠盐一水合物,n-(5-(5-水杨酰基)二钠盐一水合物)氯水杨酸基- 5-氨基己酸,正-(5-水杨酰基)-8-氨基辛酸二钠盐结晶乙醇溶剂化物,正-(5-氯水杨酰基)-5-氨基己酸二钠盐形式iii,辛酸八烷基酯盐正-(5-水杨酰基)- 8-氨基辛酸二钠,n-(5-水杨酰基)-8-氨基辛酸二钠盐一水合物,药物组合物,制备形式i(5-水杨酰基)-8-氨基辛酸的正二钠盐的方法,n -(5-水杨酰基)-8-氨基辛酸二钠盐单乙醇溶剂化物,制备5-乙酰氨基辛酸八丁酸酯的方法,iv形式的正-(5-水杨酰基)-8-氨基辛酸二钠盐和混合物制备方法形式i和iv的n-(5-水杨酰基)-8-氨基辛酸二钠盐

摘要

N- (5-CHLOROSALICYL) -5-AMINOCAPROIC ACID DISSODIC SALT, CRYSTALINE N- (5-SALICILOIL) -8-ANINOCAPRONIC ACID DISSODIC SALT, N- (5-CHLOROSALICYL) -5-AMINOCAPROIC CHLOROSALYCILOIL, N- (5-SALYCYLOIL) -8-AMINOCAPRILIC ACID DISSODIC SALT, N-(5-CHLOROSALYCILOIL) -5-AMINOCHYLROCOTIC DISSODIC SALT OF N- (5-SALICILOIL) -8-AMINOCAPRILIC ACID, CRYSTALLINE MONSHYDRATE OF N- (5-SALICILOIL) -8-AMINOCAPRILIC ACID, PHARMACEUTICAL COMPOSITION, PROCESS FOR PREPARING FORM I OF DISSODIC AC 5-SALICILOIL) -8-AMINOCAPRILIC, PROCESS TO PREPARE A MONOETHANOL SOLVATE OF N- (5-SALICILOIL) -8-AMINOCAPRILIC ACID DISSODIC SALT, PROCESS TO PREPARE 5-CNAC OCTAHYDRATE FOR PROCESS FOR IV N- (5-SALICILOIL) -8-AMINOCAPRILIC ACID DISSODIC SALT AND PROCESS FOR PREPARING A MIXTURE OF THE IV AND FORMS OF SALT N- (5-SALICYL) -8-AMINOCAPRYLIC ACID DISSODIC. The present invention relates to crystalline polymorphic forms of the N- (5-salicyloyl) -8-aminocaprylic acid disodium salt, pharmaceutical compositions containing them, methods for preparing them, and methods for facilitating the release of active agents with same.
机译:N-(5-氯水杨酸)-5-氨基己二酸二盐盐,结晶N-(5-水杨酸)-8-苯甲酸四氢二盐盐,N-(5-氯水杨酸)-5-氨基己二酸三氯盐盐,N-(5-水杨酸)-8-N-(5-水杨酸)-8-酰胺酸的N-(5-氯水杨酸)-5-氨基戊酸分散盐,N-(5-水杨酸)-8-酰胺酸的结晶单甲酸盐酸,药物成分,制备分散型AC 5-唾液酸-8-氨基己酸的晶型I的方法,制备N-(5-唾液醛)-8-氨基癸酸分散酸盐的单醇溶剂的过程,制备5-CN的过程ⅣN-(5-水杨基)-8-氨基癸酸二分散盐的邻苯二甲酸盐的制备工艺以及制备N-(5-水杨酸)-8-氨癸酸二盐盐的IV和形式的混合物的方法。本发明涉及N-(5-水杨酰基)-8-氨基辛酸二钠盐的结晶多晶型物,包含它们的药物组合物,其制备方法,以及用其促进活性剂释放的方法。

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