首页> 外国专利> NEW TRIAZOLE DERIVATIVES 4,3-a PYRIDINE, METHOD OF THEIR PRODUCTION, THEIR APPLICATION AS A MEDICINE, PHARMACEUTICAL COMPOSITIONS AND A NEW APPLICATION, IN PARTICULAR AS INHIBITORS

NEW TRIAZOLE DERIVATIVES 4,3-a PYRIDINE, METHOD OF THEIR PRODUCTION, THEIR APPLICATION AS A MEDICINE, PHARMACEUTICAL COMPOSITIONS AND A NEW APPLICATION, IN PARTICULAR AS INHIBITORS

机译:新的三唑衍生物[4,3-a]吡啶,其生产方法,其在药物中的应用,药物组合物和新的应用,特别是作为抑制剂

摘要

The invention relates to new products of formula (I) in which Ra is H, Hal, aryl or heteroaryl, optionally substituted; Rb is H, Re, —COORc, —CO — Rc or —CO — NRcRd; where Rc is alkyl, cycloalkyl, heterocycloalkyl, aryl and heteroaryl, possibly all substituted; Rd is H, alk or cycloalkyl; moreover, these products are in any isomeric forms and in the form of salts, as medicines, in particular MET inhibitors.
机译:本发明涉及式(I)的新产物,其中R a是H,Hal,芳基或杂芳基,任选地被取代; Rb为H,Re,-COORc,-CO-Rc或-CO-NRcRd;其中Rc是烷基,环烷基,杂环烷基,芳基和杂芳基,可能全部被取代; Rd是H,烷基或环烷基;此外,这些产物为药物的任何异构体形式和盐形式,特别是MET抑制剂。

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