Compounds derived from 4H, 6h 5 oxa - - - - - 2,3,10b triaza benzo e azulenes, V1a Receptor Antagonists; extraction process; Pharmaceutical composition that contains it; use in Pathological States such as dysmenorrhea, hypertension, Liver cirrhosis, nephrotic syndrome, anxiety, among others.

摘要

The present invention provides 4H,6H-5-oxa-2,3,10b-triaza-benzo[e]azulenes of the formula wherein R1 and R2 are as defined herein and which act as V1a receptor modulators, and in particular as V1a receptor antagonists, their manufacture, pharmaceutical compositions containing them and their use as medicaments.