首页> 外国专利> Endothelin-1 mRNA expression increase inhibitor, stem cell growth factor mRNA expression increase inhibitor, basic fibroblast growth factor mRNA expression increase inhibitor, and proopiomelanocortin mRNA expression increase inhibitor

Endothelin-1 mRNA expression increase inhibitor, stem cell growth factor mRNA expression increase inhibitor, basic fibroblast growth factor mRNA expression increase inhibitor, and proopiomelanocortin mRNA expression increase inhibitor

机译:内皮素-1mRNA表达增加抑制剂,干细胞生长因子mRNA表达增加抑制剂,碱性成纤维细胞生长因子mRNA表达增加抑制剂和原皮黑素皮质素mRNA表达增加抑制剂

摘要

PPROBLEM TO BE SOLVED: To provide an endothelin-1 mRNA-expression elevation inhibitor, an SCF mRNA-expression elevation inhibitor, a bFGF mRNA-expression elevation inhibitor and a POMC mRNA-expression elevation inhibitor, each comprising a flavone compound having inhibitory actions against elevations of endothelin-1 mRNA expression, SCF mRNA expression, bFGF mRNA expression and POMC mRNA expression as an active ingredient. PSOLUTION: The endothelin-1 mRNA-expression elevation inhibitor, the SCF mRNA-expression elevation inhibitor, the bFGF mRNA-expression elevation inhibitor and the POMC mRNA-expression elevation inhibitor each comprises a carambolaflavone compound as the active ingredient. PCOPYRIGHT: (C)2011,JPO&INPIT
机译:解决的问题:提供内皮素-1mRNA表达升高抑制剂,SCFmRNA表达升高抑制剂,bFGF mRNA表达升高抑制剂和POMCmRNA表达升高抑制剂,它们各自包含具有以下特征的黄酮化合物:对内皮素-1 mRNA表达,SCF mRNA表达,bFGF mRNA表达和POMC mRNA表达的升高具有抑制作用。

解决方案:内皮素-1 mRNA表达升高抑制剂,SCF mRNA表达升高抑制剂,bFGF mRNA表达升高抑制剂和POMC mRNA表达升高抑制剂各自包含杨桃黄酮化合物作为有效成分。

版权:(C)2011,日本特许厅&INPIT

著录项

  • 公开/公告号JP5634087B2

    专利类型

  • 公开/公告日2014-12-03

    原文格式PDF

  • 申请/专利权人 丸善製薬株式会社;

    申请/专利号JP20100057264

  • 发明设计人 木曽 昭典;屋敷 圭子;新穂 大介;

    申请日2010-03-15

  • 分类号A61K31/7048;A61K8/49;A61Q19/02;A61P43;A61P17;A61P13/12;A61P9;A61P17/16;A61P9/10;A61P9/12;C07D407/14;

  • 国家 JP

  • 入库时间 2022-08-21 15:27:45

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