首页> 外国专利> IMIDAZOTHIADIAZOLE DERIVATIVES AS PROTEASE ACTIVATED RECEPTOR 4 (PAR4) INHIBITORS FOR TREATING PLATELET AGGREGATION.

IMIDAZOTHIADIAZOLE DERIVATIVES AS PROTEASE ACTIVATED RECEPTOR 4 (PAR4) INHIBITORS FOR TREATING PLATELET AGGREGATION.

机译:咪唑并噻唑衍生物作为蛋白酶活化的受体4(PAR4)抑制剂用于治疗血小板聚集。

摘要

The present invention provides imidazothiadiazole compounds of Formula (I) wherein A, B, D, Rx, R1, R2, R3, X1, X2 and s are as defined herein, or a stereoisomer, tautomer, pharmaceutically acceptable salt or solvate form thereof, wherein all of the variables are as defined herein. These compounds are inhibitors of platelet aggregation and thus can be used as medicaments.
机译:本发明提供了式(I)的咪唑并噻二唑化合物,其中A,B,D,Rx,R1,R2,R3,X1,X2和s如本文所定义,或其立体异构体,互变异构体,药学上可接受的盐或溶剂化物形式,其中所有变量均如本文所定义。这些化合物是血小板聚集的抑制剂,因此可以用作药物。

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