首页> 外国专利> Combination of methyl ((1S) - 1 - ((2S) - 2 - (5 - (4 '- (2 - ((2S) - 2 - (Methoxycarbonyl) amino) - 3 - metilbutanoil) - 2 - pirrolidinil) - 1H imidazole - 5 - il) - 4 - bifenilil) - 1H imidazole - il - 2 - 1 - pirrolidinil) carbonyl) - 2-methylpropyl) carbamate (daclatasvir) and N - (tert Butoxycarbonyl) - 3 - methyl - l-valyl - (4R) - 7 - (4 - (4 - methoxy - chlorine - 1 - ISO Quinolinil Oxy) - N - ((1R,(2S) - 1 - (cyclopropylsulfonyl) Carbamoyl) - 2 - vinilciclopropil) - L - (prolinamida asunaprevir).

Combination of methyl ((1S) - 1 - ((2S) - 2 - (5 - (4 '- (2 - ((2S) - 2 - (Methoxycarbonyl) amino) - 3 - metilbutanoil) - 2 - pirrolidinil) - 1H imidazole - 5 - il) - 4 - bifenilil) - 1H imidazole - il - 2 - 1 - pirrolidinil) carbonyl) - 2-methylpropyl) carbamate (daclatasvir) and N - (tert Butoxycarbonyl) - 3 - methyl - l-valyl - (4R) - 7 - (4 - (4 - methoxy - chlorine - 1 - ISO Quinolinil Oxy) - N - ((1R,(2S) - 1 - (cyclopropylsulfonyl) Carbamoyl) - 2 - vinilciclopropil) - L - (prolinamida asunaprevir).

机译:甲基((1S)-1-((2S)-2-(5-(4'-(2-((2S)-2-(甲氧羰基)氨基))-3-甲硝丁油)-2-吡咯烷腈)-的组合1H咪唑-5-il)-4-联苯丙胺)-1H咪唑-il-2-1-吡咯烷基(羰基)-2-甲基丙基)氨基甲酸酯(daclatasvir)和N-(叔丁氧羰基)-3-甲基-l-戊基-(4R)-7-(4-(4--甲氧基-氯-1-ISO喹啉基氧基)-N-((1R,(2S)-1-(环丙基磺酰基)氨基甲酰基)-2-乙烯基氯丙醇)-L-( prolinamida asunaprevir)。

摘要

Referring to a composition comprising a compound of formula (i), which is Methyl ((1S) - 1 - ((2S) - 2 - (5 - (4 '- (2 - ((2S) - 2 - (Methoxycarbonyl) amino) - 3 - metilbutanoil) - 2 - pirrolidinil) - 1H imidazole - 5 - il) - 4 - bifenilil) - 1H imidazole - il - 2 - 1 - pirrolidinil) carbonyl) - 2-methylpropyl) carbamate (daclatasvir) and co Mpuesto of formula (ii),Which is (tert Butoxycarbonyl) - 3 - methyl - l-valyl - (4R) - 4 - (7 - (4 - methoxy - chlorine - 1 - isoquinolinil Oxy) - N - ((1R, 2S) - 1 - ((cyclopropylsulfonyl) Carbamoyl) - 2 - vinilciclopropil) - L - prolinamida (asunaprevir). The composition can inhibit the hepatitis C virus (HCV), being useful in the treatment of Type C Hepatitis
机译:涉及包含式(i)化合物的组合物,该化合物为甲基((1S)-1-((2S)-2-(5-(4'-(2-((2S)-2-(甲氧羰基)氨基)-3-甲氨蝶呤油)-2-吡咯烷腈)-1H咪唑-5-il)-4-联苯丙胺)-1H咪唑-il-2-1-吡咯烷腈)(羰基)-2-甲基丙基)氨基甲酸酯(达克拉斯韦)和式(ii)的化合物,其中为(叔丁氧羰基)-3-甲基-1-戊基-(4R)-4-(7-(4-甲氧基-氯-1-异喹啉基氧基)-N-(((1R, 2S)-1-(((环丙基磺酰基)氨基甲酰基)-2-乙烯基吡咯烷酮)-L-prolinamida(asunaprevir)。该组合物可抑制丙型肝炎病毒(HCV),可用于治疗C型肝炎

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