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NEW CRYSTAL FORM OF SODIUM-GLUCOSE CO-TRANSPORTER INHIBITOR PROCESSES FOR PREPARATION AND USE THEREOF

机译:钠-葡萄糖共转运体抑制剂的新晶体形式及其制备和使用

摘要

The present disclosure relates to novel crystalline forms of a sodium-glucose co-transporter inhibitor drug (Sotagliflozin), processes for preparation and use thereof. The present disclosure also relates to pharmaceutical composition comprises novel crystalline forms of Sotagliflozin and use of novel crystalline forms and pharmaceutical composition of Sotagliflozin for preparing drugs for treating diseases. The crystalline forms provided by the present disclosure have advantages of good stability, relatively low hygroscopicity, suitability for process development and post-treatment, simple processes for preparation, low cost, and has significant value for future drug optimization and development.
机译:本公开涉及钠-葡萄糖共转运蛋白抑制剂药物(Sotagliflozin)的新型晶体形式,其制备方法和用途。本公开还涉及包含索格列净的新型晶体形式的药物组合物,以及索格列净的新型晶体形式和药物组合物在制备用于治疗疾病的药物中的用途。本发明提供的结晶形式具有稳定性好,吸湿性相对较低,适合于工艺开发和后处理,制备工艺简单,成本低的优点,并且对于未来药物的优化和开发具有重要的价值。

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