Synthesis and Biological Activities of α-Amino Acylamines Derivatives Containing Furan and Pyridine Ring

摘要

In order to find better herbicidal activity and fungicidal activity of α-amino acid derivatives, we introduced furan rings and pyridyl groups to seven different α-amino acids to form a series of 14 novel α-amino acylamines derivatives via dicyclohexylcarbodiimide/4-dimethylaminopyridine(DCC/DMAP) coupling method. The structures of all the compounds prepared were confirmed by IR, LC/MS, 1H NMR, and elemental analysis. The herbicidal and fungicidal results show that some compounds containing glycine and valine substrate have good activities.