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机译:基于N-酰基-N-烷基磺酰胺弹头,使用小分子共价抑制剂增强抑制细胞中的蛋白质 - 蛋白质相互作用
Department of Synthetic Chemistry and Biological Chemistry Graduate School of Engineering Kyoto University Kyoto 615-8510 Japan;
Department of Synthetic Chemistry and Biological Chemistry Graduate School of Engineering Kyoto University Kyoto 615-8510 Japan;
Department of Synthetic Chemistry and Biological Chemistry Graduate School of Engineering Kyoto University Kyoto 615-8510 Japan;
Department of Synthetic Chemistry and Biological Chemistry Graduate School of Engineering Kyoto University Kyoto 615-8510 Japan;
School of Chemistry and Astbury Centre for Structural Molecular Biology University of Leeds Leeds LS2 9JT United Kingdom;
School of Chemistry and Astbury Centre for Structural Molecular Biology University of Leeds Leeds LS2 9JT United Kingdom;
Department of Synthetic Chemistry and Biological Chemistry Graduate School of Engineering Kyoto University Kyoto 615-8510 Japan ERATO (Exploratory Research for Advanced Technology JST) Tokyo 102-0075 Japan;
机译:基于药理学的HIV-1整合酶和细胞辅因子LEDGF / p75之间的蛋白质相互作用的小分子抑制剂的发现。
机译:靶向与共价小分子抑制剂的蛋白质 - 蛋白质相互作用
机译:基于热点的蛋白质-蛋白质相互作用小分子抑制剂设计
机译:共价抑制蛋白质 - 蛋白质相互作用(1):基于N-酰基-N-烷基磺酰胺(NASA)弹头的共价抑制剂的发育
机译:蛋白质-蛋白质相互作用的小分子抑制剂的合理设计:在致癌c-Myc / Max相互作用中的应用。
机译:使用配体定向的N-酰基-N-烷基磺酰胺对细胞内天然蛋白进行快速标记和共价抑制
机译:基于甲烷基烷基磺酰胺弹头的小分子共价抑制剂,增强了细胞中蛋白质蛋白相互作用的抑制